Potent and selective non-competitive mGluR5 antagonist that displays inverse agonist properties, blocks mGluR5 constitutive activity in vitro (IC50=87nM). Acts at an allosteric modulatory site shared with MPEP (Prod. No. ALX-550-368) and binds mGluR5 wit
Molecular Weight:
266.7
Purity:
98% (1H-NMR)
CAS Number:
[57653-26-6]
Formula:
C11H11ClN4O2
Target:
mGluR5
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