A classic L-type Ca2+ channel blocker (IC50=75nM) which can also inhibit T-type Ca2+ channels (IC50=244nM). It is a novel inhibitor of drug transport by p-glycoprotein (both stereoisomers are equipotent at inhibition of p-glycoprotein).
Molecular Weight:
646.2
Purity:
95% (TLC)
CAS Number:
[119934-51-9]
Formula:
C36H39N3O6 . HCl
Target:
Calcium channel (L-type), P-glycoprotein
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