BCTC is a potent and selective inhibitor of capsaicin-induced (IC50=35 nM) and acid-induced (IC50=6 nM) VR1 activation. It displays analgesic activity in rat models of inflammatory and neuropathic pain. TRPV1 antagonist.
Molecular Weight:
372.9
Purity:
98% (HPLC)
CAS Number:
[393514-24-4]
Formula:
C20H25ClN4O
Target:
TRPV1
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