Binds to calmodulin, inhibiting Ca2+-calmodulin-regulated enzyme activity. It inhibits the Ca2+/calmodulin-induced activation of myosin light chain kinase in a concentration dependent manner (IC50=25 µM). Cell permeable.
Molecular Weight:
377.3
Purity:
98% (TLC)
CAS Number:
[61714-27-0]
Formula:
C16H21ClN2O2S . HCl
Target:
Calmodulin, MLCK
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