Chemical Name: (S)-2-(3-((1-(4-Methoxybenzoyl)-2-methyl-5-(trifluoromethoxy)-1H-indol-3-yl)methyl)phenoxy)propanoic acid
PPARgamma partial agonist
Molecular Weight:
527.49
Purity:
98% by TLC, NMR (Conforms)
Form:
White solid
CAS Number:
[393794-17-7]
Formula:
C28H24F3NO6
Application Notes:
Displays high affinity for PPARgamma with excellent anti-diabetic activity in mice but poor PPARgamma agonist activity in transcription and adipogenesis assays. Highly effective (30 nM) at blocking Cdk5-mediated phosphorylation of PPARgamma. Cell permeable.
* VAT and and shipping costs not included. Errors and price changes excepted