Varenicline, CAS [[249296-44-4]]

Product Overview

• Article Name: Varenicline, CAS [[249296-44-4]]
• Biozol Catalog Number: MCE-HY-10019
• Supplier Catalog Number: HY-10019
• Alternative Catalog Number: MCE-HY-10019-5MG,MCE-HY-10019-25MG,MCE-HY-10019-10MMX1ML,MCE-HY-10019-50MG,MCE-HY-10019-100MG,MCE-HY-10019-10MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: CP 526555

Product Description

Varenicline (CP 526555) is an orally active partial agonist of alpha4beta2 nicotinic acetylcholine receptor (alpha4beta2 nAChR, IC50 = 250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of alpha6beta2 nAChR and a full agonist of alpha7beta2 nAChR. Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation[1][2][3][4][5].

Product Properties

• Molecular Weight: 211.268
• Purity: 99.92
• CAS Number: [249296-44-4]
• Formula: C13H13N3
• Target: nAChR

Application Notes

• Application Notes: Reference compound