GSK6853, a chemical probe, is a potent and selective inhibitor of the BRPF1 bromodomain. GSK6853 shows excellent BRPF1 potency (pKd = 9.5) and greater than 1600-fold selectivity over all other bromodomains[1].
Molecular Weight:
409.48
Purity:
99.89
CAS Number:
[1910124-24-1]
Formula:
C22H27N5O3
Target:
Epigenetic Reader Domain
Application Notes:
Reference compound
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