TCS-OX2-29 is a potent, high affinities and selective orexin-2 receptor (OX2R) antagonist with an IC50 value of 40 nM and a pKI value of 7.5. TCS-OX2-29 displays ~250-fold selectivity for OX2 over OX1[1][2].
Molecular Weight:
397.51
Purity:
99.55
CAS Number:
[372523-75-6]
Formula:
C23H31N3O3
Target:
Orexin Receptor (OX Receptor)
Application Notes:
Reference compound
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