GSK484 hydrochloride is a selective and reversible peptidylarginine deiminase 4 (PAD4) inhibitor. GSK484 hydrochloride demonstrates high affinity binding to PAD4 with IC50s of 50 nM in the absence of Calcium. In the presence of 2 mM Calcium, notably lower potency (250 nM) is observed.
Molecular Weight:
510.03
Purity:
99.48
CAS Number:
[1652591-81-5]
Formula:
C27H32ClN5O3
Target:
Protein Arginine Deiminase
Application Notes:
MCE Product type: Reference compound
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