GKI-1, CAS [[2444764-03-6]]

Product Overview

• Article Name: GKI-1, CAS [[2444764-03-6]]
• Biozol Catalog Number: MCE-HY-100521
• Supplier Catalog Number: HY-100521
• Alternative Catalog Number: MCE-HY-100521-10MG,MCE-HY-100521-5MG,MCE-HY-100521-10MMX1ML
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

GKI-1 is a Greatwall (GWL) kinase inhibitor with IC50s of 4.9 and 2.5 µM against hGWLFL and hGWL-KinDom, respectively. GKI-1 robustly inhibits ROCK1 with an IC50 of 11 µM, but only weakly affected PKA[1].

Product Properties

• Molecular Weight: 269.73
• Purity: 99.96
• CAS Number: [2444764-03-6]
• Formula: C15H12ClN3
• Target: ROCK

Application Notes

• Application Notes: MCE Product type: Reference compound