Lesogaberan (napadisylate), CAS [[477956-38-0]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-10061A
Supplier Catalog Number:
HY-10061A
Alternative Catalog Number:
MCE-HY-10061A-1UNIT
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Alternative Names:
AZD-3355 (napadisylate)
Lesogaberan (AZD-3355) napadisylate is a potent and selective GABAB receptor agonist with an EC50 of 8.6 nM for human recombinant GABAB receptors. The affinity (Kis) of Lesogaberan napadisylate for rat GABAB and GABAA receptors, as measured by displacement of [3H]GABA binding in brain membranes: 5.1 nM and 1.4 µM, respectively. Lesogaberan napadisylate inhibits transient lower esophageal sphincter relaxation through a peripheral mode of action[1].
Molecular Weight:
349.31
CAS Number:
[477956-38-0]
Formula:
C13H17FNO5PS
Target:
GABA Receptor
Application Notes:
MCE Product type: Reference compound1
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