Didesmethyl cariprazine, CAS [[839712-25-3]]

Product Overview

• Article Name: Didesmethyl cariprazine, CAS [[839712-25-3]]
• Biozol Catalog Number: MCE-HY-100658
• Supplier Catalog Number: HY-100658
• Alternative Catalog Number: MCE-HY-100658-5MG,MCE-HY-100658-10MG,MCE-HY-100658-25MG,MCE-HY-100658-50MG,MCE-HY-100658-100MG,MCE-HY-100658-10MMX1ML
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

Didesmethyl cariprazine is an orally active, BBB-permeable metabolite of Cariprazine (HY-14763). Didesmethyl cariprazine is a partial agonist at the D2 and D3 receptors, full agonist at the 5-HT1A receptor, and antagonist at the human 5-HT2B receptor (Ki: 1.41 nM (human D2L), 0.056 nM (human D3), 1.7 nM (human 5-HT1A), 0.52 nM (human 5-HT2B)). Didesmethyl cariprazine dose-dependently inhibits the spontaneous activity of rat midbrain dopaminergic neurons[1][2].

Product Properties

• Molecular Weight: 399.36
• Purity: 99.63
• CAS Number: [839712-25-3]
• Formula: C19H28Cl2N4O
• Target: 5-HT Receptor,Dopamine Receptor

Application Notes

• Application Notes: Reference compound