RS 39604 is a potent, selective, and orally active 5-HT4 receptor antagonist with a pKi of 9.1 in guinea pig striatal membranes. RS 39604 displays a low affinity (pKi1A, 5-HT2C, 5-HT3, alpha1c, D1, D2, M1, M2, AT1, B1 and opioid mu receptors and moderate affinity for delta1, (pKi=6.8) and delta2 (pKi=7.8) sites[1].
Molecular Weight:
590.56
Purity:
98
CAS Number:
[167710-87-4]
Formula:
C26H37Cl2N3O6S
Target:
5-HT Receptor
Application Notes:
MCE Product type: Reference compound1
* VAT and and shipping costs not included. Errors and price changes excepted