RS-102221 is a selective 5-HT2C receptor antagonist (Ki=10 nM). RS-102221 shows nearly 100-fold selectivity for the 5-HT2C receptor as compared to the 5-HT2A and 5-HT2B receptors. RS-102221 can promote the differentiation of new nerve cells. RS-102221 increases food-intake and weight-gain in rats[1][2].
Molecular Weight:
612.62
CAS Number:
[185376-97-0]
Formula:
C27H31F3N4O7S
Target:
5-HT Receptor
Application Notes:
MCE Product type: Reference compound
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