Dot1L-IN-1 TFA is a highly potent and selective Dot1L inhibitor with a Ki of 2 pM and an IC50 of 50=3 nM), as well as the activity of the HoxA9 promoter (IC50=17 nM) in HeLa and Molm-13 cells, respectively[1].
Molecular Weight:
760.23
Purity:
99.59
Formula:
C34H37ClF3N9O4S
Target:
Histone Methyltransferase
Application Notes:
MCE Product type: Reference compound
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