Gefapixant is an orally active and potent purinergic P2X3 receptor (P2X3R) antagonist, with IC50 values of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. Gefapixant can be used for the research of chronic cough and knee osteoarthritis[1][2][3].
Molecular Weight:
353.40
Purity:
99.93
CAS Number:
[1015787-98-0]
Formula:
C14H19N5O4S
Target:
P2X Receptor
Application Notes:
MCE Product type: Reference compound
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