Gefapixant (citrate), CAS [[2310299-91-1]]

Catalog Number: MCE-HY-101588A
Article Name: Gefapixant (citrate), CAS [[2310299-91-1]]
Biozol Catalog Number: MCE-HY-101588A
Supplier Catalog Number: HY-101588A
Alternative Catalog Number: MCE-HY-101588A-5MG,MCE-HY-101588A-10MG,MCE-HY-101588A-25MG,MCE-HY-101588A-100MG,MCE-HY-101588A-10MMX1ML,MCE-HY-101588A-50MG
Manufacturer: MedchemExpress
Category: Biochemikalien
Alternative Names: MK-7264 (citrate), AF-219 (citrate)
Gefapixant citrate is an orally active and potent purinergic P2X3 receptor (P2X3R) antagonist, with IC50 values of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. Gefapixant citrate can be used for the research of chronic cough and knee osteoarthritis[1][2][3].
Molecular Weight: 545.52
Purity: 99.23
CAS Number: [2310299-91-1]
Formula: C20H27N5O11S
Target: P2X Receptor
Application Notes: MCE Product type: Reference compound