Gefapixant (Standard) is the analytical standard of Gefapixant. This product is intended for research and analytical applications. Gefapixant is an orally active and potent purinergic P2X3 receptor (P2X3R) antagonist, with IC50 values of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors. Gefapixant can be used for the research of chronic cough and knee osteoarthritis[1][2][3].
Molecular Weight:
353.40
CAS Number:
[1015787-98-0]
Formula:
C14H19N5O4S
Target:
P2X Receptor,Reference Standards
Application Notes:
MCE Product type: Reference Standards
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