RP-001 is a picomolar short-acting S1P1 (EDG1) selective agonist, with an EC50 of 9 pM. RP-00 induces internalization and polyubiquitination of S1P1. RP-001 has little activity on S1P2-S1P4 and only moderate affinity for S1P5[1].
Molecular Weight:
432.47
CAS Number:
[1306761-53-4]
Formula:
C24H24N4O4
Target:
LPL Receptor
Application Notes:
MCE Product type: Reference compound
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