Ruboxistaurin-d6 (hydrochloride) is the deuterium labeled Ruboxistaurin hydrochloride. Ruboxistaurin (LY333531) hydrochloride is an orally active, selective PKC beta inhibitor (Ki=2 nM). Ruboxistaurin hydrochloride exhibits ATP dependent competitive inhibition of PKC beta I with an IC50 of 4.7 nM. Ruboxistaurin hydrochloride inhibits PKC beta II with an IC50 of 5.9 nM[1][2].
Molecular Weight:
511.04
CAS Number:
[1794767-04-6]
Formula:
C28H23D6ClN4O3
Target:
Isotope-Labeled Compounds,PKC
Application Notes:
MCE Product type: Isotope-Labeled Compounds
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