SB 243213 hydrochloride is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 hydrochloride shows greater than a 100-fold selectivity over a wide range of neurotransmitter receptors, enzymes and ion channels. SB 243213 hydrochloride has improved anxiolytic profile and has the potential for schizophrenia and motor disorders[1].
Molecular Weight:
464.87
Purity:
98.84
CAS Number:
[200940-23-4]
Formula:
C22H20ClF3N4O2
Target:
5-HT Receptor
Application Notes:
MCE Product type: Reference compound
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