SB 243213 is an orally active, selective and high-affinity 5-HT2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 shows greater than a 100-fold selectivity over a wide range of neurotransmitter receptors, enzymes and ion channels. SB 243213 has improved anxiolytic profile and has the potential for schizophrenia and motor disorders[1].
Molecular Weight:
428.41
Purity:
99.4400
CAS Number:
[200940-22-3]
Formula:
C22H19F3N4O2
Target:
5-HT Receptor
Application Notes:
MCE Product type: Reference compound
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