NAS-181 (dimesylate), CAS [[1217474-40-2]]

Product Overview

• Article Name: NAS-181 (dimesylate), CAS [[1217474-40-2]]
• Biozol Catalog Number: MCE-HY-103156
• Supplier Catalog Number: HY-103156
• Alternative Catalog Number: MCE-HY-103156-25MG,MCE-HY-103156-10MMX1ML,MCE-HY-103156-100MG,MCE-HY-103156-5MG,MCE-HY-103156-10MG,MCE-HY-103156-50MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

NAS181 is a potent and selective antagonist of rat 5-HT1B receptor, with a Ki of 47 nM. NAS181 shows 13-fold selectivity for r5-HT1B over bovine 5-HT1B receptor (Ki=630 nM). NAS181 increases the 5-HT turnover and the synaptic concentration of 5-HT by inhibiting terminal r5-HT1B autoreceptors[1][2].

Product Properties

• Molecular Weight: 538.63
• Purity: 96.37
• CAS Number: [1217474-40-2]
• Formula: C21H34N2O10S2
• Target: 5-HT Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound