PSB-10 hydrochloride is a potent and selective antagonist of human adenosine A3 receptor (A3AR), with a Ki of 0.44 nM. PSB-10 hydrochloride shows more than 800-fold selectivity for hA3 over rA1, rA2A, hA1, hA2A and hA2B receptors (Ki=805, 6040, 1700, 2700, 30000 nM, respectively). PSB-10 hydrochloride produces thermal hyperalgesia in mice[1][2].
Molecular Weight:
435.14
CAS Number:
[591771-91-4]
Formula:
C16H15Cl4N5O
Target:
Adenosine Receptor
Application Notes:
MCE Product type: Reference compound
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