Azepexole (B-HT 933) dihydrochloride is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for alpha2A-, alpha2B- and alpha2C-adrenoceptor subtypes, resepctively[1]. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC50= 78.72 nM)[2].
Molecular Weight:
254.16
CAS Number:
[36067-72-8]
Formula:
C9H17Cl2N3O
Target:
Adrenergic Receptor
Application Notes:
MCE Product type: Reference compound
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