LE 300 is a potent and selective dopamine D1-like receptor antagonist with Kis of 1.9 nM and 7.5 nM in CHO cell membranes expressing human dopamine D1 and D5 receptors, respectively. LE 300 is an antagonist of the 5-HT2A receptor with a pA2 of 8.32 in a rat tail artery assay[1][2].
Molecular Weight:
290.40
Purity:
98.5
CAS Number:
[274694-98-3]
Formula:
C20H22N2
Target:
5-HT Receptor,Dopamine Receptor
Application Notes:
Reference compound
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