G-36 is a cell-permeable nonsteroidal antagonist of the G protein-coupled estrogen receptor (GPER/GPR30), which selectively inhibits estrogen-mediated PI3K activation through GPER, rather than Eralpha. G-36 also inhibits estrogen-mediated calcium mobilization (IC50=112 nM). G-36 is promising for research in the field of cancer[1][2].
Molecular Weight:
412.32
Purity:
99.35
CAS Number:
[1392487-51-2]
Formula:
C22H22BrNO2
Target:
Estrogen Receptor/ERR
Application Notes:
MCE Product type: Reference compound
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