Y134 is a selective and orally active oestrogen receptor (ER) modulator (SERM), exhibits potent antagonist activity at ERalpha and ERbeta. Y134 shows 121.1-fold selectivity for ERalpha (Ki=0.09 nM) over ERbeta (Ki=11.31 nM). Y134 inhibits oestrogen-stimulated proliferation of ER-positive human breast cancer cells[1].
Molecular Weight:
472.60
Purity:
99.67
CAS Number:
[849662-80-2]
Formula:
C28H28N2O3S
Target:
Estrogen Receptor/ERR
Application Notes:
MCE Product type: Reference compound
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