NNC-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1) with IC50 values of 0.04, 0.38, 171, 1700, 349, 622 µM for human GAT-1, rat GAT-1, rGAT-2, hGAT-3, rGAT-3, hBGT-3, respectively. NNC-711 has anticonvulsant and analgesic effect in vivo and exhibits cognition-enhancing activity[1][2][3][4][5].
Molecular Weight:
386.87
Purity:
99.76
CAS Number:
[145645-62-1]
Formula:
C21H23ClN2O3
Target:
GABA Receptor
Application Notes:
MCE Product type: Reference compound
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