CI-966 (hydrochloride), CAS [[110283-66-4]]

Product Overview

• Article Name: CI-966 (hydrochloride), CAS [[110283-66-4]]
• Biozol Catalog Number: MCE-HY-103534
• Supplier Catalog Number: HY-103534
• Alternative Catalog Number: MCE-HY-103534-10MMX1ML,MCE-HY-103534-5MG,MCE-HY-103534-50MG,MCE-HY-103534-10MG,MCE-HY-103534-100MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

CI-966 hydrochloride is a potent, selective, orally active and brain-penetrant inhibitor of the GABA transporter GAT-1, with IC50s of 0.26 µM and 1.2 µM for hGAT-1, rGAT-1, respectively. CI-966 hydrochloride shows more than 200-fold selectivity over GAT-2, GAT-3, and BGT-3. CI-966 hydrochloride exhibits anticonvulsant and neuroprotective activities[1][2][3].

Product Properties

• Molecular Weight: 509.87
• Purity: 99.60
• CAS Number: [110283-66-4]
• Formula: C23H22ClF6NO3
• Target: GABA Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound