YM-202074 (fumarate), CAS [[299900-84-8]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-103556
Supplier Catalog Number:
HY-103556
Alternative Catalog Number:
MCE-HY-103556-1MG,MCE-HY-103556-5MG
Manufacturer:
MedchemExpress
Category:
Biochemikalien
YM-202074 fumarate is a selective, allosteric metabotropic glutamate receptor type 1 (mGluR1) antagonist with high affinity. YM-202074 fumarate binds to the allosteric site of rat mGluR1 with a Ki of 4.8 nM. YM-202074 fumarate also inhibits mGluR1-mediated inositol phosphate production in rat cerebellar granule cells with an IC50 of 8.6 nM. YM-202074 fumarate has potent neuroprotective effects in transient MCA (tMCA) occlusion rat models[1].
Molecular Weight:
1177.34
CAS Number:
[299900-84-8]
Formula:
C56H72N8O16S2
Target:
mGluR
Application Notes:
MCE Product type: Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted