YM-202074 (fumarate), CAS [[299900-84-8]] Preis auf Anfrage

Catalog Number: MCE-HY-103556
Article Name: YM-202074 (fumarate), CAS [[299900-84-8]] Preis auf Anfrage
Biozol Catalog Number: MCE-HY-103556
Supplier Catalog Number: HY-103556
Alternative Catalog Number: MCE-HY-103556-1MG,MCE-HY-103556-5MG
Manufacturer: MedchemExpress
Category: Biochemikalien
YM-202074 fumarate is a selective, allosteric metabotropic glutamate receptor type 1 (mGluR1) antagonist with high affinity. YM-202074 fumarate binds to the allosteric site of rat mGluR1 with a Ki of 4.8 nM. YM-202074 fumarate also inhibits mGluR1-mediated inositol phosphate production in rat cerebellar granule cells with an IC50 of 8.6 nM. YM-202074 fumarate has potent neuroprotective effects in transient MCA (tMCA) occlusion rat models[1].
Molecular Weight: 1177.34
CAS Number: [299900-84-8]
Formula: C56H72N8O16S2
Target: mGluR
Application Notes: MCE Product type: Reference compound