Theliatinib (tartrate), CAS [[2413487-72-4]] Preis auf Anfrage
Biozol Catalog Number:
MCE-HY-104066A
Supplier Catalog Number:
HY-104066A
Alternative Catalog Number:
MCE-HY-104066A-1UNIT
Manufacturer:
MedchemExpress
Category:
Biochemikalien
Alternative Names:
Xiliertinib (tartrate), HMPL-309 (tartrate)
Theliatinib (Xiliertinib) tartrate is a potent, ATP-competitive, orally active and highly selective EGFR inhibitor with a Ki of 0.05 nM and an IC50 of 3 nM. Theliatinib has an IC50 of 22 nM for EGFR T790M/L858R mutant. Theliatinib shows >50-fold selectivity for EGFR than other kinases[1]. Theliatinib (tartrate) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
Molecular Weight:
592.60
CAS Number:
[2413487-72-4]
Formula:
C29H32N6O8
Target:
EGFR
Application Notes:
MCE Product type: Reference compound
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