Lerisetron is a potent 5-HT3 antagonists and possess high-affinity binding for the 5-HT3 receptors with pKi value of 9.2. Lerisetron has a potent ability to inhibit the 5-HT-evoked reflex bradycardia in urethane-anesthetized rats[1].
Molecular Weight:
292.39
Purity:
99.69
CAS Number:
[143257-98-1]
Formula:
C18H20N4
Target:
5-HT Receptor
Application Notes:
MCE Product type: Reference compound
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