Zaldaride maleate (CGS-9343B) is a potent, orally active and selective inhibitor of calmodulin. Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity, with an IC50 of 3.3 nM[1][2]. Zaldaride maleate prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+ and K+ currents in PC12 cells and inhibits nAChR[3].
Molecular Weight:
544.60
Purity:
99.7
CAS Number:
[109826-27-9]
Formula:
C30H32N4O6
Target:
Calmodulin
Application Notes:
MCE Product type: Reference compound
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