FK888 is a potent, selective, and high affinity dipeptide NK1 receptor antagonist. FK888 displaces [3H]-SP binding with a Ki value of 0.69 nM and 0.45 microM. FK888 also inhibits SP-induced airway oedema in guinea-pig after both intravenous and oral administration[1].
Molecular Weight:
588.70
CAS Number:
[138449-07-7]
Formula:
C36H36N4O4
Target:
Neurokinin Receptor
Application Notes:
MCE Product type: Reference compound
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