CI-988 hemihydrate (PD134308) is a potent, selective and orally active CCK2R (cholecystokinin 2 receptor) antagonist with an IC50 of 1.7 nM for mouse cortex CCK2. CI-988 hemihydrate shows >1600-fold selectivity for CCK2 over CCK1 receptor. CI-988 hemihydrate has anxiolytic and anti-tumor effects[1][2][3].
Molecular Weight:
623.74
Purity:
99
Formula:
C35H42N4O6.1/2H2O
Target:
Cholecystokinin Receptor
Application Notes:
MCE Product type: Reference compound
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