GSK1904529A is a potent, selective, orally active, and ATP-competitive inhibitor of insulin-like growth factor-1 receptor (IGF-1R) and insulin receptor (IR), with IC50s of 27 and 25 nM, respectively. GSK1904529A shows poor activity (IC50>1 µM) in 45 other serine/threonine and tyrosine kinases. GSK1904529A exhibits anti-tumor activity[1][2].
Molecular Weight:
851.96
Purity:
99.03
CAS Number:
[1089283-49-7]
Formula:
C44H47F2N9O5S
Target:
Apoptosis,IGF-1R,Insulin Receptor
Application Notes:
MCE Product type: Reference compound1
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