TP-9201 is a platelet glycoprotein (GP) IIb/IIIa receptor antagonist. TP-9201 inhibits the interaction between GPIIb/IIIa and fibrinogen, thereby suppressing platelet aggregation. TP-9201 exhibits similar inhibitory activity on adenosine diphosphate (ADP) (HY-W010918)-induced platelet aggregation in humans, baboons, and dogs (IC50 = 1-3 µM), while showing lower activity in rabbits (IC50 = 45 µM) and rats (IC50 = 20 µM). TP-9201can be used in studies related to the prevention of rethrombosis after arterial thrombolysis[1].
Molecular Weight:
1136.26
CAS Number:
[138297-15-1]
Formula:
C45H69N17O14S2
Target:
P-glycoprotein
Application Notes:
MCE Product type: Reference compound
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