Spiradoline (U-62066), an arylacetamide, is a selective kappa opioid receptor (KOR) agonist with a Ki of 8.6 nM in guinea pig. The Ki values of Spiradoline for µ and delta receptors are 252 nM and 9400 nM, respectively. Spiradoline has potent diuretic, analgesic, antiarrythmic, antitussive, neuroprotective properties and easily penetrates the blood-brain barrier[1][2].
Molecular Weight:
425.39
CAS Number:
[87151-85-7]
Formula:
C22H30Cl2N2O2
Target:
Opioid Receptor
Application Notes:
MCE Product type: Reference compound
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