L-365260 is an orally active and selective antagonist of non-peptide gastrin and brain cholecystokinin receptor (CCK-B), with Kis of 1.9 nM and 2.0 nM, respectively. L-365260 interacts in a stereoselective and competitive manner with guinea pig stomach gastrin and brain CCK receptors. L-365260 can enhance Morphine analgesia and prevents Morphine tolerance[1][2][3].
Molecular Weight:
398.46
Purity:
99.85
CAS Number:
[118101-09-0]
Formula:
C24H22N4O2
Target:
Cholecystokinin Receptor
Application Notes:
MCE Product type: Reference compound
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