ROS 234 is a potent H3 antagonist, with a pKB of 9.46 for Guinea-pig ileum H3-receptor, a pKi of 8.90 for Rat cerebral cortex H3-receptor, and a ED50 of 19.12 mg/kg (ip) in ex vivo of Rat cerebral cortex. ROS 234 diaplays poor central access[1][2].
Molecular Weight:
241.29
CAS Number:
[184576-87-2]
Formula:
C13H15N5
Target:
Histamine Receptor
Application Notes:
MCE Product type: Reference compound
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