VU 0365114 is a selective mAChR M5 positive allosteric modulator, with an EC50 of 2.7 µM, and >30 µM for M1, M2, M3 and M4 receptors. VU 0365114 increases insulin secretion stimulated by ACh in human beta-cells[1][2][3].
Molecular Weight:
397.35
Purity:
99.41
CAS Number:
[1208222-39-2]
Formula:
C22H14F3NO3
Target:
mAChR
Application Notes:
MCE Product type: Reference compound1
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