3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, with IC50s are 0.28, 0.30 and 31.6 nM for halpha4beta4, halpha4beta2, and halpha7-nACh, respectively. 3-Bromocytisine (3-Br-cytisine) shows different effects on high (HS) and low (LS) ACh sensitivity alpha4beta2 nAChRs with EC50s are 8 and 50 nM, respectively[1][2].
Molecular Weight:
269.14
Purity:
99.90
CAS Number:
[207390-14-5]
Formula:
C11H13BrN2O
Target:
nAChR
Application Notes:
MCE Product type: Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted