MRS2365 is a potent and selective P2Y1 receptor (EC50=0.4 nM) /[35S]GTPgammaS binding/beta-arrestin 2 recruitment agonist with an EC50 of 0.4 nM. MRS2365 relieves mechanical allodynia and increases mechanical sensitivity. MRS2365 shows little agonist or antagonist activity at the P2Y12 or P2Y13 receptors[1][2][3][4].
Molecular Weight:
483.33
CAS Number:
[436847-09-5]
Formula:
C13H19N5O9P2S
Target:
Arrestin,P2Y Receptor
Application Notes:
MCE Product type: Reference compound
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