CCG258208 (GRK2-IN-1) is a potent and selective GRK2 (G protein-coupled receptor kinase 2) inhibitor (IC50=30 nM) while maintaining 230-fold selectivity over GRK5 (IC50=7.09 µM) and more than 2500-fold selectivity over GRK1 (IC50=87.3 µM), PKA, and ROCK1. CCG258208 can be used in heart failure research[1].
Molecular Weight:
452.48
CAS Number:
[2055990-90-2]
Formula:
C24H25FN4O4
Target:
G Protein-coupled Receptor Kinase (GRK)
Application Notes:
MCE Product type: Reference compound
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