Irdabisant, CAS [[1005402-19-6]]

Product Overview

• Article Name: Irdabisant, CAS [[1005402-19-6]]
• Biozol Catalog Number: MCE-HY-109968
• Supplier Catalog Number: HY-109968
• Alternative Catalog Number: MCE-HY-109968-10MG,MCE-HY-109968-500MG,MCE-HY-109968-25MG,MCE-HY-109968-100MG,MCE-HY-109968-50MG,MCE-HY-109968-10MMX1ML,MCE-HY-109968-250MG,MCE-HY-109968-5MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: CEP-26401

Product Description

Irdabisant (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant histamine H3 receptor (H3R) inverse agonist/inverse agonist with Ki values of 7.2 nM and 2.0 nM for rat H3R and human H3R, respectively. Irdabisant has relatively low inhibitory activity against hERG current with an IC50 of 13.8 µM. Irdabisant has cognition-enhancing and wake-promoting activities in the rat social recognition model. Irdabisant can be used to research schizophrenia or cognitive impairment[1][2].

Product Properties

• Molecular Weight: 313.39
• Purity: 99.58
• CAS Number: [1005402-19-6]
• Formula: C18H23N3O2
• Target: Histamine Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound