ETP-45658 is a potent PI3K inhibitor, with IC50s of 22.0 nM, 39.8 nM, 129.0 nM and 717.3 nM for PI3Kalpha, PI3Kdelta, PI3Kbeta and PI3Kgamma, respectively. ETP-45658 also can inhibit DNA-PK (IC50=70.6 nM) and mTOR (IC50=152.0 nM). ETP-45658 can be used for the research of cancer[1][2].
Molecular Weight:
311.34
Purity:
98.97
CAS Number:
[1198357-79-7]
Formula:
C16H17N5O2
Target:
DNA-PK,mTOR,PI3K
Application Notes:
MCE Product type: Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted