Eplivanserin (SR-46349) hemifumarate is a potent, selective and orally active 5-HT2A receptor antagonist, with an IC50 of 5.8 nM in rat cortical membrane, and a Kd of 1.14 nM. Eplivanserin hemifumarate displays >20-fold selectivity more selective for 5-HT2A than 5-HT2B and 5-HT2C[1][2].
Molecular Weight:
386.43
Purity:
99.10
CAS Number:
[130580-02-8]
Formula:
C19H21FN2O2.1/2C4H4O4
Target:
5-HT Receptor
Application Notes:
MCE Product type: Reference compound1
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