PQ-69 is a potent and selective adenosine A1 receptor antagonist with inverse agonist activity. PQ-69 binds to hA1 receptor with a Ki value of 0.96 nM, is 217-fold more selective compared with hA2A receptors (Ki=208 nM) and >1,000-fold selectivity over hA3 receptor (Ki >100 µM). PQ-69 can be used for the research of renal dysfunction[1].
Molecular Weight:
350.39
CAS Number:
[910045-32-8]
Formula:
C20H19FN4O
Target:
Adenosine Receptor
Application Notes:
MCE Product type: Reference compound1
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