NVS-CECR2-1, CAS [[1992047-61-6]]

Catalog Number: MCE-HY-110374
Article Name: NVS-CECR2-1, CAS [[1992047-61-6]]
Biozol Catalog Number: MCE-HY-110374
Supplier Catalog Number: HY-110374
Alternative Catalog Number: MCE-HY-110374-5MG,MCE-HY-110374-25MG,MCE-HY-110374-10MMX1ML,MCE-HY-110374-50MG,MCE-HY-110374-10MG,MCE-HY-110374-100MG
Manufacturer: MedchemExpress
Category: Biochemikalien
NVS-CECR2-1, a non-BET family Bromodomain (BRD) inhibitor, is a potent and selective cat eye syndrome chromosome region, candidate 2 (CECR2) inhibitor. NVS-CECR2-1 binds to CECR2 BRD with high affinity (IC50=47 nM, KD=80 nM). NVS-CECR2-1 exhibits cytotoxic activity and induces apoptosis against various cancer cells by targeting CECR2 as well as via CECR2-independent mechanism[1]. NVS-CECR2-1 is a chemical probe.
Molecular Weight: 495.68
Purity: 99.40
CAS Number: [1992047-61-6]
Formula: C27H37N5O2S
Target: Apoptosis,Epigenetic Reader Domain
Application Notes: MCE Product type: Reference compound